SCHEMBL8005145

SCHEMBL8005145

COc1cc(OC)c2c(N)cc(-c3cc(C(C)C)on3)nc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
ALDH1A1 P00352 6/20 0.37
HPGD P15428 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 3/20 0.37
GBA1 P04062 1/20 0.37
S1PR1 P21453 1/20 0.33
RET P07949 2/20 0.33
MEN1 O00255 2/20 0.32
CYP1A2 P05177 2/20 0.32
MAPK1 P28482 2/20 0.32
CYP2C19 P33261 2/20 0.32
KMT2A Q03164 2/20 0.32
ELANE P08246 2/20 0.32
CYP3A4 P08684 2/20 0.32
MAPT P10636 2/20 0.32
PDGFRB P09619 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15216108 0.86 PDE3B (0.41) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL15216092 0.85 PDE3B (0.38) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL8008296 0.79 ALDH1A1 (0.40) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL7993475 0.77 PDE3B (0.37) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL577253 0.76 SMN1; SMN2 (0.37) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL7995961 0.75 SLC2A1 (0.43) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL8002114 0.74 CYP1A1 (0.37) PDE3BPDE3AALDH1A1HPGDSMN1; SMN2
SCHEMBL7992813 0.73 PDE10A (0.32) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL8007996 0.72 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL7995957 0.69 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed