SCHEMBL8005489

SCHEMBL8005489

C=CCO[C@H]1CCCN(C(N)=O)C1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.35
PDE4B Q07343 3/20 0.34
CYP11B2 P19099 2/20 0.33
EPHX2 P34913 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 1/20 0.32
LMNA P02545 2/20 0.31
CPN1 P15169 1/20 0.31
CPB2 Q96IY4 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8012170 1.00 TAAR1 (0.35) TAAR1PDE4BCYP11B2EPHX2ALDH1A1
SCHEMBL1072300 0.86 TAAR1 (0.38) TAAR1EPHX2ALDH1A1MAPK1LMNA
SCHEMBL18669321 0.86 TAAR1 (0.38) TAAR1EPHX2ALDH1A1MAPK1LMNA
SCHEMBL17099260 0.81 GRM5 (0.40) TAAR1PDE4BEPHX2ALDH1A1LMNA
SCHEMBL8010277 0.79 MEN1 (0.49) PDE4BALDH1A1MEN1KMT2A
SCHEMBL20477490 0.79 MEN1 (0.49) PDE4BALDH1A1MEN1KMT2A
SCHEMBL8005512 0.79 KMT2A (0.36) TAAR1EPHX2LMNASMN1; SMN2MEN1
SCHEMBL5793762 0.76 EPHX2 (0.35) EPHX2
SCHEMBL16530276 0.76 EPHX2 (0.35) EPHX2
SCHEMBL31618749 0.75 HPGD (0.46) PDE4BALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086982-B1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2018-08-29 EP disclosed
US-9738661-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-22 US disclosed
US-20150266897-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2015-09-24 US disclosed
WO-2009108507-A1 THERAPEUTIC COMPOUNDS MERCK & CO., INC. (US) 2009-09-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150266897-A1 HCV NS3 Protease Inhibitors HAVCR2, GTF3C3, CTSC TAAR1 4659/4885PDE4B 3619/4885CYP11B2 1721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.