SCHEMBL8008235

SCHEMBL8008235

Cn1cnc2c(Cc3ccccc3)nc(N)nc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.62
MPO P05164 1/20 0.49
CDK2 P24941 3/20 0.46
CCNB1 P14635 2/20 0.46
CCNE1 P24864 2/20 0.46
LTB4R Q15722 1/20 0.46
CYP1A2 P05177 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HIF1A Q16665 1/20 0.45
PHLPP2 Q6ZVD8 1/20 0.45
CCNA2 P20248 2/20 0.44
CCNA1 P78396 2/20 0.44
KDM4E B2RXH2 1/20 0.44
CCNB2 O95067 1/20 0.44
CCNE2 O96020 1/20 0.44
GAA P10253 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24021885 0.79 CDK1 (0.53) CDK1CDK2CCNB1CCNE1CYP1A2
SCHEMBL2153011 0.78 CYP2C19 (0.47) CDK1MPOCYP1A2ALDH1A1CYP3A4
SCHEMBL3209666 0.78 CDK1 (0.60) CDK1MPOCDK2CCNB1CCNE1
SCHEMBL13521265 0.78 CDK1 (0.50) CDK1CDK2CCNB1CCNE1CYP1A2
SCHEMBL8648457 0.78 CYP2C19 (0.49) MPOCYP1A2ALDH1A1CYP3A4CYP2C9
SCHEMBL14612509 0.77 CDK1 (0.51) CDK1CDK2CCNB1CCNE1CYP1A2
SCHEMBL8647716 0.77 CDK1 (0.52) CDK1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7999866 0.77 CDK1 (1.00) CDK1CDK2CCNB1CCNE1CYP1A2
SCHEMBL13866472 0.77 CDK1 (0.62) CDK1CDK2CCNB1CCNE1CYP1A2
SCHEMBL6266942 0.76 CYP2C19 (0.45) CDK1MPOCDK2CCNB1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000033657-A1 METHOD TO IDENTIFY REGULATORS OF CDK ACTIVITY CROPDESIGN N.V. (BE) 2000-06-15 WO disclosed