SCHEMBL8008329

SCHEMBL8008329

COc1ccc(-c2nnn(C)n2)cc1CCCc1nnc(C)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.42
ALDH1A1 P00352 4/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 2/20 0.39
ACLY P53396 1/20 0.39
LMNA P02545 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MAPK1 P28482 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
LRRK2 Q5S007 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGD P15428 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8013904 0.97 TACR1 (0.42) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL8009641 0.88 TACR1 (0.39) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL8009206 0.82 TRPV1 (0.41) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL8005781 0.81 ALDH1A1 (0.37) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL10293072 0.78 MAPT (0.43) ALDH1A1ATMMAPTLMNAL3MBTL1
SCHEMBL8009821 0.77 MAPT (0.38) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL8010506 0.77 TACR1 (0.41) TACR1ALDH1A1ATMMAPTACLY
SCHEMBL8009636 0.76 SPHK2 (0.38) ALDH1A1MAPTLMNAL3MBTL1MAPK1
SCHEMBL10260401 0.76 MAPT (0.39) ALDH1A1ATMMAPTLMNAL3MBTL1
SCHEMBL10292902 0.76 MAPT (0.43) ALDH1A1ATMMAPTLMNATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed