SCHEMBL8008499

SCHEMBL8008499

O=C(CCc1ccccc1)c1ccc(OCCO)cc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.68
RAB9A P51151 1/20 0.68
GAA P10253 1/20 0.62
FFAR1 O14842 4/20 0.59
ABCB1 P08183 7/20 0.55
MAPT P10636 2/20 0.54
HRH3 Q9Y5N1 1/20 0.53
ALDH1A1 P00352 1/20 0.53
RECQL P46063 1/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.51
FFAR4 Q5NUL3 1/20 0.51
EGFR P00533 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697972 0.94 GAA (0.62) NPC1RAB9AGAAFFAR1ABCB1
SCHEMBL1557011 0.84 FFAR1 (0.71) NPC1RAB9AGAAFFAR1MAPT
SCHEMBL23877665 0.82 MAPT (0.61) NPC1GAAMAPTHRH3ALDH1A1
Dietifen SCHEMBL2109562 0.81 NPC1 (0.62) NPC1RAB9AFFAR1ABCB1MAPT
SCHEMBL8008112 0.81 NPC1 (0.62) NPC1RAB9AFFAR1ABCB1MAPT
SCHEMBL1304210 0.81 NPC1 (1.00) NPC1RAB9AABCB1MAPTALDH1A1
SCHEMBL9081465 0.81 NPC1 (0.76) NPC1RAB9AFFAR1ABCB1MAPT
SCHEMBL19160273 0.81 GAA (0.60) NPC1RAB9AGAAFFAR1MAPT
SCHEMBL128056 0.81 GAA (0.75) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL11403932 0.81 FFAR1 (0.57) NPC1RAB9AFFAR1MAPTHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP claimed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO claimed
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
US-5834506-A TREATMENT OF HIV, AIDS; ANTIVIRAL ACTIVITY IMPROVED BY JUDICIOUS PLACEMENT OF POLAR SUBSTITUENTS WARNER-LAMBERT COMPANY (US) 1998-11-10 US disclosed