SCHEMBL8009033

SCHEMBL8009033

COC(C)C1CC[C@H]2[C@@H]3C(C)CC4OC(=O)C=C[C@]4(C)[C@@H]3CC[C@]12C

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 9/20 0.47
SRD5A2 P31213 8/20 0.47
GPBAR1 Q8TDU6 2/20 0.35
NR1H4 Q96RI1 1/20 0.35
FNTA P49354 2/20 0.34
FNTB P49356 2/20 0.34
SHBG P04278 3/20 0.33
NR3C1 P04150 1/20 0.32
CYP17A1 P05093 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009030 1.00 SRD5A1 (0.47) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL8003369 0.90 SRD5A1 (0.49) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL8003366 0.90 SRD5A1 (0.49) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL8002701 0.83 SRD5A1 (0.44) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL8002703 0.83 SRD5A1 (0.44) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL7993713 0.83 SRD5A1 (0.69) SRD5A1SRD5A2FNTAFNTB
SCHEMBL8316920 0.82 SRD5A1 (0.47) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL7993711 0.82 SRD5A1 (0.47) SRD5A1SRD5A2GPBAR1NR1H4FNTA
SCHEMBL8319303 0.82 SRD5A1 (0.33) SRD5A1SRD5A2
SCHEMBL8319307 0.82 SRD5A1 (0.33) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858455-A4 4-OXA AND 4-THIA STEROIDS MERCK & CO INC (US) 2000-04-12 EP claimed
EP-0858455-A1 4-OXA AND 4-THIA STEROIDS Merck & Co., Inc. (US) 1998-08-19 EP claimed
US-5777134-A 4-oxa and 4-thia steriods MERCK & CO., INC. (US) 1998-07-07 US claimed
WO-1997015564-A1 4-OXA AND 4-THIA STEROIDS MERCK & CO., INC. (US) 1997-05-01 WO claimed
US-5998464-A 4-Oxa and 4-thia steroids MERCK & CO., INC. (US) 1999-12-07 US disclosed
US-5932559-A Treatment of hyperandrogenic conditions MERCK & CO., INC. (US) 1999-08-03 US disclosed
US-5777134-A 4-oxa and 4-thia steriods MERCK & CO., INC. (US) 1998-07-07 US disclosed
US-5756480-A Treatment of hyperandrogenic conditions MERCK & CO., INC. (US) 1998-05-26 US disclosed
WO-1997015305-A1 TREATMENT OF HYPERANDROGENIC CONDITIONS MERCK & CO., INC. (US) 1997-05-01 WO disclosed