SCHEMBL8316920

SCHEMBL8316920

COC(C)[C@H]1CC[C@H]2[C@@H]3[C@@H](C)C[C@H]4SC(=O)C=C[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 9/20 0.47
SRD5A2 P31213 8/20 0.47
NR1H4 Q96RI1 4/20 0.35
GPBAR1 Q8TDU6 3/20 0.35
FNTA P49354 2/20 0.34
FNTB P49356 2/20 0.34
SHBG P04278 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993711 1.00 SRD5A1 (0.47) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL8005881 0.90 SRD5A1 (0.49) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL7994159 0.90 SRD5A1 (0.49) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL8003605 0.83 SRD5A1 (0.44) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL8531614 0.83 SRD5A1 (0.44) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL8323073 0.83 SRD5A1 (0.44) SRD5A1SRD5A2NR1H4GPBAR1FNTA
SCHEMBL8003079 0.83 SRD5A1 (0.69) SRD5A1SRD5A2FNTAFNTB
SCHEMBL8019380 0.82 SRD5A1 (0.33) SRD5A1SRD5A2
SCHEMBL8019377 0.82 SRD5A1 (0.33) SRD5A1SRD5A2
SCHEMBL8009033 0.82 SRD5A1 (0.47) SRD5A1SRD5A2NR1H4GPBAR1FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998464-A 4-Oxa and 4-thia steroids MERCK & CO., INC. (US) 1999-12-07 US claimed
US-5998464-A 4-Oxa and 4-thia steroids MERCK & CO., INC. (US) 1999-12-07 US disclosed
US-5932559-A Treatment of hyperandrogenic conditions MERCK & CO., INC. (US) 1999-08-03 US disclosed
US-5777134-A 4-oxa and 4-thia steriods MERCK & CO., INC. (US) 1998-07-07 US disclosed
US-5756480-A Treatment of hyperandrogenic conditions MERCK & CO., INC. (US) 1998-05-26 US disclosed
WO-1997015305-A1 TREATMENT OF HYPERANDROGENIC CONDITIONS MERCK & CO., INC. (US) 1997-05-01 WO disclosed