SCHEMBL8009191

SCHEMBL8009191

BrC(Br)Oc1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP2C19 P33261 2/20 0.49
KDM4E B2RXH2 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 2/20 0.48
CYP2C9 P11712 1/20 0.48
HTR1B P28222 4/20 0.46
SLC6A4 P31645 10/20 0.45
SLC6A2 P23975 9/20 0.45
SLC6A3 Q01959 2/20 0.44
NR2E1 Q9Y466 1/20 0.43
KCNA3 P22001 1/20 0.43
HPGD P15428 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HTR1D P28221 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27613071 0.83 HTR1B (0.47) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL11577421 0.82 KDM4E (0.52) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL1356983 0.79 HTR1B (0.47) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL30942689 0.79 SLC6A4 (0.47) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL4982131 0.78 CYP1A2 (0.56) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL13971022 0.78 KDM4E (0.49) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL10344137 0.78 KDM4E (0.49) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL6831487 0.78 HTR1B (0.50) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL5072033 0.78 SLC6A2 (0.53) CYP1A2CYP2C19KDM4EMEN1KMT2A
SCHEMBL9329809 0.77 CYP1A2 (0.49) CYP1A2CYP2C19KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973714-A2 PRODUCTION OF RACEMIC 2-(6-METHOXY-2-NAPHTHYL)PROPIONIC ACID OR PRECURSORS THEREOF ALBEMARLE CORPORATION (US) 2000-01-26 EP disclosed
EP-0937021-A1 PRODUCTION OF NABUMETONE OR PRECURSORS THEREOF ALBEMARLE CORPORATION (US) 1999-08-25 EP disclosed
US-5907069-A METHYLATION OF 6-BROMO-2-NAPHTHOL WITH METHYL BROMIDE OR METHYL CHLORIDE AND RECOVERING NABUMETONE ALBEMARLE CORPORATION (US) 1999-05-25 US disclosed
US-5840996-A Production of brominated methoxynaphthalene compounds ALBEMARLE CORPORATION (US) 1998-11-24 US disclosed
WO-1998050334-A1 PRODUCTION OF BROMINATED METHOXYNAPHTHALENE COMPOUNDS ALBEMARLE CORPORATION (US) 1998-11-12 WO disclosed
US-5792886-A METHYLATION OF 6-BROMO-2-NAPHTHOL WITH METHYL BROMIDE TO 2-BROMO-6-METHOXYNAPHTHALENE; FORMING GRIGNARD; REACTING WITH A LOWER ALKYL 2-BROMOPROPIONATE ALBEMARLE CORPORATION (US) 1998-08-11 US disclosed
WO-1998030528-A2 PRODUCTION OF RACEMIC 2-(6-METHOXY-2-NAPHTHYL)PROPIONIC ACID OR PRECURSORS THEREOF ALBEMARLE CORPORATION (US) 1998-07-16 WO disclosed
US-5756851-A Production of nabumetone or precursors thereof ALBEMARLE CORPORATION (US) 1998-05-26 US disclosed
WO-1998017616-A1 PRODUCTION OF NABUMETONE OR PRECURSORS THEREOF ALBEMARLE CORPORATION (US) 1998-04-30 WO disclosed