SCHEMBL8009741

SCHEMBL8009741

CN(C)CCNCCc1cccnc1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.70
CHRNB2 P17787 3/20 0.54
CHRNA4 P43681 3/20 0.54
SIGMAR1 Q99720 1/20 0.49
CHRM2 P08172 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP2A6 P11509 1/20 0.45
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
HTR5A P47898 1/20 0.44
ALDH1A1 P00352 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16606311 0.86 CYP1A2 (0.63) CHRNA7CHRM2CYP1A2CYP2D6TDP1
SCHEMBL8001649 0.85 CYP1A2 (0.65) CHRNA7CHRNB2CHRNA4CHRM2CYP1A2
SCHEMBL8363021 0.83 CHRNA7 (1.00) CHRNA7CHRNB2CHRNA4CHRM2CYP1A2
SCHEMBL30772178 0.83 CHRNA7 (1.00) CHRNA7CHRNB2CHRNA4CHRM2CYP1A2
SCHEMBL22762150 0.81 TDP1 (0.61) CHRNA7CHRNB2CHRNA4SIGMAR1CHRM2
SCHEMBL10282657 0.80 TDP1 (0.58) CHRNA7CHRNB2CHRNA4CHRM2CYP1A2
SCHEMBL11846860 0.80 CHRNA7 (0.79) CHRNA7CHRNB2CHRNA4SIGMAR1TDP1
SCHEMBL10858987 0.80 CYP1A2 (0.55) CHRNA7CHRM2CYP1A2CYP2D6TDP1
SCHEMBL11411955 0.79 KCNH2 (0.65) SIGMAR1
SCHEMBL8111184 0.79 CHRNB2 (0.47) CHRNA7CHRNB2CHRNA4SIGMAR1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057318-A ANTAGONISTS OF PLATELET ACTIVATING FACTOR ACETHER SANOFI (FR) 2000-05-02 US disclosed
US-5470855-A Anticoagulants SANOFI (FR) 1995-11-28 US disclosed