SCHEMBL8009926

SCHEMBL8009926

COc1ccncc1C[C@@H](N)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
TSPO P30536 2/20 0.41
OPRK1 P41145 2/20 0.41
CYP3A4 P08684 2/20 0.41
SLC7A5 Q01650 1/20 0.41
USP2 O75604 2/20 0.41
HIF1A Q16665 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
BLM P54132 2/20 0.41
PMP22 Q01453 2/20 0.41
KMT2A Q03164 2/20 0.41
RGS12 O14924 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32661890 0.80 MAPT (0.39) CA12CA1CA2CA9TSPO
SCHEMBL28741574 0.80 GRIA1 (0.48) HSD17B10CYP3A4SLC7A5USP2HIF1A
Hydrochloric Acid SCHEMBL31407596 0.79 MAPT (0.39) CA12CA1CA2CA9TSPO
SCHEMBL2263341 0.78 HSD17B10 (0.49) HSD17B10CYP3A4SLC7A5USP2HIF1A
SCHEMBL155235 0.78 NOS3 (0.55) SLC7A5HIF1AKDM4EMEN1LMNA
SCHEMBL155234 0.78 NOS3 (0.55) SLC7A5HIF1AKDM4EMEN1LMNA
SCHEMBL4595466 0.78 NOS3 (0.55) SLC7A5HIF1AKDM4EMEN1LMNA
SCHEMBL29750308 0.78 NOS3 (0.55) SLC7A5HIF1AKDM4EMEN1LMNA
SCHEMBL13957557 0.77 GRIA1 (0.48) HSD17B10CYP3A4SLC7A5USP2HIF1A
SCHEMBL30759485 0.77 HSD17B10 (0.47) HSD17B10CYP3A4SLC7A5USP2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850316-A4 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIV HAWAII (US) 2000-08-23 EP disclosed
EP-0850316-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1998-07-01 EP disclosed
WO-1997008334-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1997-03-06 WO disclosed