SCHEMBL8010147

SCHEMBL8010147

COc1ccc(C2N=NN(C)N2)cc1/C=C/CCCc1csc(C)n1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
HTR2B P41595 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
ALDH1A1 P00352 2/20 0.31
RAB9A P51151 1/20 0.31
HCRTR2 O43614 1/20 0.31
CHEK1 O14757 1/20 0.31
CYP1A2 P05177 1/20 0.31
SLC5A7 Q9GZV3 1/20 0.31
METAP2 P50579 1/20 0.31
NTRK1 P04629 1/20 0.30
CSF1R P07333 1/20 0.30
NTRK2 Q16620 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8005862 0.97 HTR2A (0.32) HTR2AHTR2CSLC6A4HTR2BL3MBTL1
SCHEMBL8009623 0.89 HTR2A (0.34) HTR2AHTR2CSLC6A4HTR2BL3MBTL1
SCHEMBL8000552 0.82
SCHEMBL8010341 0.74 TRPV1 (0.38) L3MBTL1ALDH1A1RAB9ACHEK1NTRK1
SCHEMBL7999092 0.72 ALDH1A1 (0.36) HTR2AHTR2CSLC6A4HTR2BL3MBTL1
SCHEMBL8012587 0.71 TRPV1 (0.40) L3MBTL1ALDH1A1RAB9ACHEK1NTRK1
SCHEMBL7998586 0.70 ALDH1A1 (0.35) L3MBTL1ALDH1A1RAB9ACYP1A2SLC5A7
SCHEMBL8010265 0.68 ALDH1A1 (0.37) L3MBTL1ALDH1A1RAB9ACHEK1NTRK1
SCHEMBL8005747 0.66 ALDH1A1 (0.37) HTR2AHTR2CSLC6A4HTR2BL3MBTL1
SCHEMBL8008233 0.63 ALDH1A1 (0.38) L3MBTL1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed