SCHEMBL8010248

SCHEMBL8010248

[c]1ccc(N(CCCc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.57
CHRM2 P08172 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
SLC6A3 Q01959 1/20 0.47
AOC3 Q16853 1/20 0.47
SIGMAR1 Q99720 4/20 0.47
KCNA3 P22001 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999176 0.83 KCNH2 (0.48) KCNH2CHRM2HTR1AADRA2ACHRM1
Bromide SCHEMBL11785438 0.82 KCNH2 (0.62) KCNH2CHRM2HTR1AADRA2ACHRM1
SCHEMBL21628965 0.81 MEN1 (0.44) KCNH2OPRM1SIGMAR1
SCHEMBL7825708 0.80 SIGMAR1 (0.53) KCNH2CHRM2HTR1AADRA2ACHRM1
SCHEMBL6999585 0.79 SIGMAR1 (0.56) KCNH2CHRM2HTR1AADRA2ACHRM1
SCHEMBL7003391 0.79 SIGMAR1 (0.56) KCNH2CHRM2HTR1AADRA2ACHRM1
SCHEMBL8001156 0.79 NPC1 (0.45) KCNH2SIGMAR1
SCHEMBL5843435 0.79 NR3C2 (0.47) KCNH2AOC3KCNA3
SCHEMBL8010122 0.78 KCNH2 (0.57) KCNH2CHRM2HTR1AADRA2ACHRM1
SCHEMBL668551 0.78 HTR2A (0.54) ADRA1ASLC6A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1066729-C Benzimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-06-06 CN disclosed
CN-1060173-C Heterocyclic compound with activity against diabetes and preparation and application of same MITSUTAKA CO LTD (JP) 2001-01-03 CN disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
CN-1157288-A Benzimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1997-08-20 CN disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
CN-1118781-A Heterocyclic compound with activity against diabetes and preparation and application of same MITSUTAKA CO LTD (JP) 1996-03-20 CN disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed