SCHEMBL8011323

SCHEMBL8011323

Oc1ccc(-c2cccc3ncccc23)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.59
CA1 P00915 2/20 0.59
CA2 P00918 2/20 0.59
CA9 Q16790 2/20 0.59
ERN1 O75460 4/20 0.52
ACVR1 Q04771 4/20 0.51
MAPT P10636 4/20 0.47
KDM4E B2RXH2 2/20 0.47
FYN P06241 1/20 0.46
BMP4 P12644 1/20 0.46
CASP1 P29466 2/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MCL1 Q07820 1/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KMT2A Q03164 2/20 0.44
COMT P21964 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27278122 0.87 BMP4 (0.57) CA12CA1CA2CA9ACVR1
SCHEMBL12074247 0.84 CA12 (0.65) CA12CA1CA2CA9ERN1
SCHEMBL4658401 0.83 CA12 (0.59) CA12CA1CA2CA9ERN1
SCHEMBL4073648 0.82 CA12 (0.59) CA12CA1CA2CA9ERN1
SCHEMBL6296099 0.82 CA12 (0.59) CA12CA1CA2CA9ERN1
SCHEMBL27737402 0.82 CA12 (0.63) CA12CA1CA2CA9ERN1
SCHEMBL12386951 0.82 CA12 (0.59) CA12CA1CA2CA9ERN1
SCHEMBL9669763 0.81 CA12 (0.58) CA12CA1CA2CA9ERN1
SCHEMBL21935175 0.81 CA1 (0.55) CA12CA1CA2CA9ERN1
SCHEMBL17334527 0.81 CA12 (0.57) CA12CA1CA2CA9ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106103417-B The derivative and preparation method thereof of 1,2- naphthoquinones KT&G生命科学公司 2019-08-06 CN disclosed
CN-105164113-B Pyrroloamide inhibitors 艾伯维公司 2018-03-02 CN disclosed
CN-106103417-A Derivant of 1,2 naphthoquinone and preparation method thereof KT&G生命科学公司 2016-11-09 CN disclosed
CN-105992759-A 1, 2-naphthoquinone derivative and preparation method thereof KT&G生命科学公司 2016-10-05 CN disclosed
CN-105164113-A Pyrroloamide inhibitors ABBVIE INC 2015-12-16 CN disclosed
CN-101541753-B 2-aminoquinolines as 5-HT(5A) receptor antagonists HOFFMANN LA ROCHE 2012-06-13 CN disclosed
CN-101516852-B Quinoline derivatives with 5-ht-binding properties HOFFMANN LA ROCHE 2011-11-16 CN disclosed
CN-101541753-A 2-Aminoquinolines as 5-HT(5A) receptor antagonists HOFFMANN LA ROCHE (CH) 2009-09-23 CN disclosed
CN-101516852-A Quinoline derivatives with 5-HT-binding properties HOFFMANN LA ROCHE (CH) 2009-08-26 CN disclosed
US-6124460-A Isoquinuclidine derivatives, method of manufacturing the same and therapeutic agents for hypercholesterolemia containing these compounds KOTOBUKI PHARMACEUTICAL CO. LTD. (JP) 2000-09-26 US disclosed