SCHEMBL8012182

SCHEMBL8012182

CCCCc1nc(-c2ccc(N)cc2)c[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 4/20 0.44
GSK3B P49841 1/20 0.43
HRH3 Q9Y5N1 2/20 0.40
HRH2 P25021 1/20 0.40
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
XDH P47989 2/20 0.36
SREBF2 Q12772 1/20 0.36
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35
KMT2A Q03164 2/20 0.35
NOS2 P35228 1/20 0.35
KEAP1 Q14145 1/20 0.34
METAP2 P50579 1/20 0.34
ASIC3 Q9UHC3 1/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016347 0.95 TLR8 (0.47) TLR8GSK3BHRH3HRH2RAB9A
SCHEMBL8012754 0.90 SREBF2 (0.41) TLR8GSK3BHRH3HRH2RAB9A
SCHEMBL13277717 0.84 GSK3B (0.43) TLR8GSK3BRAB9ASMN1; SMN2NPC1
SCHEMBL22585763 0.84 RAD52 (0.44) TLR8RAB9ASMN1; SMN2NPC1TP53
SCHEMBL6618330 0.84 GSK3B (0.44) TLR8GSK3BRAB9ASMN1; SMN2NPC1
SCHEMBL8012285 0.83 TLR8 (0.39) TLR8RAB9ASMN1; SMN2NPC1TP53
Ammonia Solution, Strong SCHEMBL27564785 0.83 GSK3B (0.43) TLR8GSK3BRAB9ASMN1; SMN2NPC1
SCHEMBL4943588 0.80 GAA (0.37) TLR8RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL6129194 0.80 TLR8 (0.45) TLR8GSK3BHRH3RAB9ANPC1
SCHEMBL17626094 0.79 GSK3B (0.41) GSK3BRAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed