SCHEMBL8012235

SCHEMBL8012235

Cc1nc(-c2cccc(NC(=C3C(=O)Nc4ccc([N+](=O)[O-])cc43)c3ccccc3)c2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
PDE4D Q08499 1/20 0.39
RIPK1 Q13546 1/20 0.39
CNR1 P21554 1/20 0.39
GSK3B P49841 2/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
CAPN9 O14815 1/20 0.38
CASP3 P42574 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.38
ALOX5 P09917 1/20 0.38
TGM2 P21980 1/20 0.38
ALDH1A1 P00352 1/20 0.37
THRB P10828 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8012232 1.00 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8013336 0.92 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8013331 0.92 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8001470 0.90 EGFR (0.39) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8010847 0.90 ABCG2 (0.43) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8010843 0.90 ABCG2 (0.43) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8001473 0.90 EGFR (0.39) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8012180 0.88 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8012183 0.88 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD
SCHEMBL8517816 0.85 EGFR (0.42) EGFRMEN1KMT2ALMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed