SCHEMBL8001470

SCHEMBL8001470

CCc1nc(-c2cccc(N/C(=C3\C(=O)Nc4ccc([N+](=O)[O-])cc43)c3ccccc3)c2)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 3/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
F2 P00734 1/20 0.38
LMNA P02545 2/20 0.37
RIPK1 Q13546 1/20 0.37
PDE4D Q08499 1/20 0.37
GSK3B P49841 1/20 0.36
MAPK1 P28482 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
CAPN9 O14815 1/20 0.36
CASP3 P42574 1/20 0.36
TGM2 P21980 1/20 0.36
BACE1 P56817 2/20 0.36
ALOX5 P09917 1/20 0.36
ACHE P22303 1/20 0.35
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001473 1.00 EGFR (0.39) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8001471 0.93 EGFR (0.40) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8001474 0.93 EGFR (0.40) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8012232 0.90 EGFR (0.42) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8012235 0.90 EGFR (0.42) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8010847 0.87 ABCG2 (0.43) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8010843 0.87 ABCG2 (0.43) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8010512 0.87 MEN1 (0.40) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8010518 0.87 MEN1 (0.40) EGFRMEN1KMT2AHPGDMAPT
SCHEMBL8012853 0.85 EGFR (0.38) EGFRMEN1KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed