Bicarbonate

Bicarbonate

SCHEMBL8017378

Cc1cc(C)c(CC(=O)C2CCC2)c(C)c1.O=C(O)O

nearest known ligand 0.45

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.40
POLB P06746 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 3/20 0.38
TAS1R3 Q7RTX0 4/20 0.37
TAS1R1 Q7RTX1 4/20 0.37
TAS1R2 Q8TE23 4/20 0.37
HRH3 Q9Y5N1 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 1/20 0.36
P2RX7 Q99572 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL8022789 0.95 EPHX2 (0.45) EPHX2NPSR1LMNAGAATAS1R3
Bicarbonate SCHEMBL8005996 0.88 EPHX2 (0.36) EPHX2POLBNPSR1LMNAGAA
Bicarbonate SCHEMBL8022729 0.87 EPHX2 (0.37) EPHX2POLBTAS1R3TAS1R1TAS1R2
Bicarbonate SCHEMBL8005963 0.85 POLB (0.36) EPHX2POLBNPSR1LMNAGAA
Bicarbonate SCHEMBL8005998 0.84 EPHX2 (0.35) EPHX2POLBNPSR1LMNAGAA
Bicarbonate SCHEMBL8015563 0.83 GRM1 (0.37) EPHX2POLBKDM4EMAPTALDH1A1
Bicarbonate SCHEMBL8019371 0.81 EPHX2 (0.34) EPHX2POLBNPSR1GAATAS1R3
Bicarbonate SCHEMBL8019208 0.81 TAS1R3 (0.42) EPHX2POLBNPSR1GAATAS1R3
Bicarbonate SCHEMBL8018120 0.80 TAS1R3 (0.34) EPHX2POLBTAS1R3TAS1R1TAS1R2
Bicarbonate SCHEMBL8021766 0.80 EPHX2 (0.34) EPHX2POLBTAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773920-B1 2-(2,4,6-TRIMETHYL PHENYL)CYCLOPENTANE-1,3-DIONE DERIVATIVES BAYER AG (DE) 2000-01-26 EP disclosed
EP-0773920-A1 2-(2,4,6-TRIMETHYL PHENYL)CYCLOPENTANE-1,3-DIONE DERIVATIVES BAYER AG (DE) 1997-05-21 EP disclosed
WO-1996003366-A1 2-(2,4,6-TRIMETHYL PHENYL)CYCLOPENTANE-1,3-DIONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1996-02-08 WO disclosed