SCHEMBL8018654

SCHEMBL8018654

CC(c1c[nH]c2ccccc12)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 2/20 0.46
TP53 P04637 2/20 0.46
CASP3 P42574 4/20 0.45
PIN1 Q13526 2/20 0.45
KMT2A Q03164 1/20 0.43
MDM2 Q00987 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6480706 1.00 MDM4 (0.46) MDM4TP53CASP3PIN1KMT2A
SCHEMBL31000753 1.00 MDM4 (0.46) MDM4TP53CASP3PIN1KMT2A
SCHEMBL5913024 1.00 MDM4 (0.46) MDM4TP53CASP3PIN1KMT2A
SCHEMBL31000751 1.00 MDM4 (0.46) MDM4TP53CASP3PIN1KMT2A
SCHEMBL6481998 1.00 MDM4 (0.46) MDM4TP53CASP3PIN1KMT2A
SCHEMBL31000614 0.87 CASP3 (0.43) MDM4TP53CASP3PIN1KMT2A
SCHEMBL31000582 0.87 FFAR1 (0.43) MDM4TP53CASP3PIN1MDM2
SCHEMBL31000535 0.85 HDAC3 (0.43) MDM4TP53CASP3PIN1KMT2A
SCHEMBL31000490 0.85 MDM4 (0.43) MDM4TP53CASP3PIN1MDM2
SCHEMBL6225058 0.84 TACR1 (0.44) PIN1KMT2AMDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063796-A HETEROCYCLIC COMPOUNDS OF PIPERIDINE MERCK & CO., INC. (US) 2000-05-16 US disclosed
US-6057338-A USEFUL IN THE TREATMENT OF DIABETES, CANCER, ACROMEGALY, RESTENOSIS, DEPRESSION, IRRITABLE BOWEL SYNDROME, PAIN AND DIABETIC RETINOPATHY MERCK & CO., INC. (US) 2000-05-02 US disclosed