SCHEMBL8019073

SCHEMBL8019073

CCN1CCN(c2nc3c(S(=O)(=O)c4cc(C)ccc4C)nnn3c3ccsc23)CC1

nearest known ligand 0.84

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 7/20 0.84
HTR6 P50406 12/20 0.81
MAPT P10636 4/20 0.61
TP53 P04637 1/20 0.60
POLB P06746 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016806 0.91 RXFP1 (1.00) RXFP1HTR6MAPTTP53POLB
SCHEMBL8028821 0.89 HTR6 (1.00) RXFP1HTR6MAPTTP53POLB
SCHEMBL8028237 0.89 HTR6 (0.85) RXFP1HTR6MAPTTP53POLB
SCHEMBL8034015 0.88 HTR6 (1.00) RXFP1HTR6MAPTTP53POLB
SCHEMBL8027276 0.85 RXFP1 (0.79) RXFP1HTR6MAPTTP53POLB
SCHEMBL8018164 0.82 HTR6 (0.83) RXFP1HTR6MAPTTP53POLB
SCHEMBL8028840 0.80 RXFP1 (0.75) RXFP1HTR6MAPTTP53
SCHEMBL8027731 0.76 HTR6 (1.00) RXFP1HTR6MAPTTP53POLB
SCHEMBL8019071 0.75 HTR6 (0.76) RXFP1HTR6MAPTPOLB
SCHEMBL15285384 0.75 HTR6 (0.84) RXFP1HTR6MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed