SCHEMBL8019231

SCHEMBL8019231

CC(C)c1ccc(C(O)C#N)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
TYR P14679 2/20 0.40
HTT P42858 2/20 0.40
ERBB2 P04626 1/20 0.38
MGLL Q99685 1/20 0.38
CYP2C9 P11712 3/20 0.36
HIF1A Q16665 2/20 0.36
ALOX5 P09917 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TRPA1 O75762 1/20 0.35
PTGS1 P23219 1/20 0.35
CACNA1C Q13936 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8020863 0.81 TSHR (0.60) TSHRESR1ESR2HTTCYP2C9
SCHEMBL197981 0.81 TSHR (0.60) TSHRESR1ESR2HIF1AALDH1A1
SCHEMBL1200882 0.81 TSHR (0.60) TSHRESR1ESR2HTTALOX5
SCHEMBL3991740 0.81 TSHR (0.60) TSHRESR1ESR2HTTALOX5
SCHEMBL6688835 0.81 TSHR (0.60) TSHRESR1ESR2HIF1AALDH1A1
SCHEMBL4328254 0.81 TSHR (0.60) TSHRESR1ESR2HIF1AALDH1A1
SCHEMBL4319988 0.78 ESR1 (0.62) TSHRESR1ESR2CYP2C9HIF1A
SCHEMBL467691 0.78 ESR1 (0.62) TSHRESR1ESR2CYP2C9HIF1A
SCHEMBL7262475 0.78 ESR1 (0.62) TSHRESR1ESR2CYP2C9HIF1A
SCHEMBL8791848 0.77 PTGS1 (0.50) TSHRESR1ESR2CYP2C9ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711836-B1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide MITSUBISHI RAYON CO (JP) 2000-02-02 EP disclosed
US-5736385-A NITRILASE OR NITRILE HYDRATASE HYDROLYSIS OF A CYANOHYDRIN WHILE AUTOMATICALLY CONTROLLING CYANOHYDRIN CONCENTRATION NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
US-5583147-A INHIBITORS OF ACYL-COENZYME A: CHOLESTEROL O-TRANSFERASE; ANTIHYPERCHOLESTEROLEMIC AND/OR ANTIATHEROSCLEROTIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-10 US disclosed
EP-0711836-A1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-05-15 EP disclosed