SCHEMBL8021048

SCHEMBL8021048

COc1cc(C2C[C@@]3(C)[C@@H](C[C@H](C)[C@@H]4[C@@H]3CC[C@]3(C)[C@@H](C(=O)O)CC[C@@H]43)NC2=O)cc(OC)c1OC

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 5/20 0.34
SRD5A2 P31213 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NR3C1 P04150 1/20 0.33
SERPINA6 P08185 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006971 0.87 SRD5A1 (0.39) SRD5A1SRD5A2
SCHEMBL8006557 0.87 SRD5A1 (0.44) SRD5A1SRD5A2
SCHEMBL8021029 0.82 SRD5A1 (0.34) SRD5A1SRD5A2NR3C1
SCHEMBL8016699 0.74 SRD5A1 (0.49) SRD5A1SRD5A2
SCHEMBL8016963 0.72 SRD5A2 (0.58) SRD5A1SRD5A2
SCHEMBL8016958 0.72 SRD5A2 (0.58) SRD5A1SRD5A2
SCHEMBL8016669 0.72 SRD5A2 (0.58) SRD5A1SRD5A2
SCHEMBL8017010 0.72 SRD5A1 (0.41) SRD5A1SRD5A2
SCHEMBL8006812 0.71 SRD5A1 (0.60) SRD5A1SRD5A2
SCHEMBL8016888 0.71 SRD5A1 (0.60) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP disclosed
US-5278159-A Steroid enzyme inhibitor MERCK & CO., INC. (US) 1994-01-11 US disclosed