SCHEMBL8021029

SCHEMBL8021029

COc1cc(C2C[C@]3(C)[C@H]4CC[C@]5(C)[C@@H](C(=O)O)CC[C@H]5[C@@H]4[C@@H](C)C[C@H]3N(C)C2=O)cc(OC)c1OC

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 2/20 0.34
SRD5A2 P31213 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR3C1 P04150 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8017010 0.87 SRD5A1 (0.41) SRD5A1SRD5A2
SCHEMBL8021048 0.82 SRD5A1 (0.34) SRD5A1SRD5A2NR3C1
SCHEMBL8023852 0.73 SRD5A1 (0.58) SRD5A1SRD5A2
SCHEMBL8023848 0.73 SRD5A1 (0.58) SRD5A1SRD5A2
SCHEMBL8006557 0.72 SRD5A1 (0.44) SRD5A1SRD5A2
SCHEMBL8016913 0.71 SRD5A1 (0.43) SRD5A1
SCHEMBL8006971 0.70 SRD5A1 (0.39) SRD5A1SRD5A2
SCHEMBL8018781 0.70 MAPT (0.38) SRD5A1ALDH1A1SMN1; SMN2
SCHEMBL8016758 0.70 MBOAT4 (0.37) NR3C1
SCHEMBL8020895 0.69 SRD5A2 (0.61) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP disclosed
US-5278159-A Steroid enzyme inhibitor MERCK & CO., INC. (US) 1994-01-11 US disclosed