SCHEMBL8022206

SCHEMBL8022206

O=C(O)C1=CNC=C(C(=O)O)C1c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
GAA P10253 5/20 0.46
KDM4E B2RXH2 4/20 0.46
GLA P06280 4/20 0.46
HPGD P15428 4/20 0.46
CASP1 P29466 3/20 0.46
CASP7 P55210 3/20 0.46
HSD17B10 Q99714 3/20 0.46
ATM Q13315 1/20 0.46
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
HTR2B P41595 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
RCE1 Q9Y256 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28854641 0.87 ALDH1A1 (0.68) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL21180531 0.82 ALDH1A1 (0.46) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL29046363 0.80 ALDH1A1 (0.73) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL26970375 0.77 ALDH1A1 (0.44) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL30512143 0.76 ALDH1A1 (0.68) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL29234076 0.73 ALDH1A1 (0.68) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL28854617 0.73 ALDH1A1 (0.68) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL30502408 0.73 GAA (0.66) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL30502405 0.73 ALDH1A1 (0.66) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL28854619 0.72 ALDH1A1 (0.67) ALDH1A1GAAKDM4EGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10167966-A None JP disclosed
JP-60038336-A None JP disclosed
CN-111362941-A Visible light preparation method of aza-tetraacetalkane compounds 北京工业大学 2020-07-03 CN disclosed
US-RE36607-E Pyrrolidine compounds and process of preparing BAYER AKTIENGESELLSCHAFT (DE) 2000-03-07 US disclosed
US-5910593-A Highly selective process for the preparation of enantiomerically pure phenylsubstituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1999-06-08 US disclosed
US-5849924-A Highly selective process for the preparation of enantiomerically pure phenyl-substituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives BAYER AKTIENGESELLSCAHFT (DE) 1998-12-15 US disclosed
JP-H10167966-A ORAL SUSTAINED RELEASE PREPARATION NIPPON CHEMIPHAR CO LTD 1998-06-23 JP disclosed
US-5700948-A CALCIUM ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 1997-12-23 US disclosed
US-5272161-A Indolesulphonamide-substituted dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1993-12-21 US disclosed
EP-0533014-A1 Indolesulfonamide substituted dihydropyridines, process for their preparation and drugs containing them BAYER AG (DE) 1993-03-24 EP disclosed
JP-S6038336-A BENZALDEHYDE DERIVATIVE AND ITS PREPARATION TEIJIN LTD 1985-02-27 JP disclosed