SCHEMBL8022559

SCHEMBL8022559

CNCCC(Oc1ccccc1C#N)c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.73
SLC6A4 P31645 14/20 0.73
CYP2D6 P10635 10/20 0.73
NOS2 P35228 7/20 0.73
KCNH2 Q12809 4/20 0.73
CYP1A2 P05177 4/20 0.66
CYP3A4 P08684 4/20 0.66
TSHR P16473 3/20 0.66
SLC6A3 Q01959 3/20 0.66
KMT2A Q03164 2/20 0.66
CHRM1 P11229 2/20 0.66
ADRA2B P18089 2/20 0.66
HTR2A P28223 2/20 0.66
HTR2C P28335 2/20 0.66
HRH1 P35367 2/20 0.66
OPRM1 P35372 2/20 0.66
DRD3 P35462 2/20 0.66
OPRK1 P41145 2/20 0.66
HTR2B P41595 2/20 0.66
KLF10 Q13118 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8022554 1.00 SLC6A2 (0.73) SLC6A2SLC6A4CYP2D6NOS2KCNH2
Hydrochloric Acid SCHEMBL6498694 0.99 SLC6A2 (0.74) SLC6A2SLC6A4CYP2D6NOS2KCNH2
Oxalic Acid SCHEMBL8011871 0.94 SLC6A2 (0.74) SLC6A2SLC6A4CYP2D6NOS2KCNH2
SCHEMBL6500144 0.86 SLC6A2 (0.77) SLC6A2SLC6A4CYP2D6NOS2KCNH2
SCHEMBL20435479 0.85 SLC6A4 (1.00) SLC6A2SLC6A4CYP2D6NOS2KCNH2
SCHEMBL6504695 0.85 SLC6A4 (0.75) SLC6A2SLC6A4CYP2D6NOS2KCNH2
SCHEMBL6493450 0.85 SLC6A4 (1.00) SLC6A2SLC6A4CYP2D6NOS2KCNH2
Hydrochloric Acid SCHEMBL6502850 0.85 SLC6A2 (0.77) SLC6A2SLC6A4CYP2D6NOS2KCNH2
Hydrochloric Acid SCHEMBL6492236 0.84 NOS2 (1.00) SLC6A2SLC6A4CYP2D6NOS2KCNH2
SCHEMBL6491411 0.84 SLC6A4 (1.00) SLC6A2SLC6A4CYP2D6NOS2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000058262-A1 STEREOSPECIFIC METHOD FOR PREPARING TOMOXETINE AND INTERMEDIATES THEREOF ELI LILLY AND COMPANY (US) 2000-10-05 WO claimed
WO-2000058262-A1 STEREOSPECIFIC METHOD FOR PREPARING TOMOXETINE AND INTERMEDIATES THEREOF ELI LILLY AND COMPANY (US) 2000-10-05 WO disclosed