SCHEMBL8025895

SCHEMBL8025895

CNC(=O)C#Cc1ccc(-n2cccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.49
ALDH1A1 P00352 3/20 0.43
AOC2 O75106 3/20 0.42
POLB P06746 3/20 0.40
NSD2 O96028 1/20 0.40
GRK2 P25098 1/20 0.40
CASP6 P55212 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
MAPT P10636 3/20 0.39
RAB9A P51151 3/20 0.39
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
LMNA P02545 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554708 0.77 NPSR1 (0.55) ALDH1A1POLBRAB9AMEN1KMT2A
SCHEMBL666992 0.74 APP (0.49) ALDH1A1POLBRAB9AMEN1KMT2A
SCHEMBL6561789 0.71 NPC1 (0.60) ACACBPOLBRAB9AMEN1KMT2A
SCHEMBL6563230 0.70 ALDH1A1 (0.43) ALDH1A1
SCHEMBL8022190 0.70 PTPN11 (0.53) ALDH1A1POLBMAPTRAB9AMEN1
SCHEMBL402534 0.69 APP (0.55) ACACBALDH1A1POLBNSD2GRK2
SCHEMBL403365 0.69 ACACB (0.49) ACACB
SCHEMBL2241437 0.67 KMT2A (0.71) ALDH1A1AOC2POLBNSD2GRK2
SCHEMBL3893087 0.67 KDM4E (0.45) ACACBALDH1A1AOC2POLBNSD2
SCHEMBL168605 0.66 ACACB (1.00) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed