SCHEMBL8026089

SCHEMBL8026089

C=C(c1ccc(C(=O)OC)cc1)c1ccc2c(c1)C(C)(OC)CCC2(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 13/20 0.60
RARB P10826 10/20 0.60
RARG P13631 9/20 0.60
RXRB P28702 7/20 0.60
RARA P10276 6/20 0.60
RXRG P48443 6/20 0.60
CYP3A4 P08684 4/20 0.55
CYP26A1 O43174 4/20 0.51
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421758 0.91 RXRA (0.72) RXRARARBRARGRXRBRARA
SCHEMBL8026151 0.89 RXRA (0.78) RXRARARBRARGRXRBRARA
SCHEMBL8026112 0.87 RARB (0.58) RXRARARBRARGRXRBRARA
SCHEMBL7896511 0.82 RXRA (0.63) RXRARARBRARGRXRBRARA
SCHEMBL9746786 0.82 RARB (0.74) RXRARARBRARGRXRBRARA
SCHEMBL8026092 0.81 RARB (0.61) RXRARARBRARGRARACYP3A4
SCHEMBL2788640 0.79 CYP3A4 (0.70) RXRARARBRARGRXRBRARA
SCHEMBL6814372 0.79 RXRA (0.49) RXRARARBRARGRXRBRARA
SCHEMBL9319204 0.77 CYP3A4 (0.67) RXRARARBRARGRXRBRARA
SCHEMBL7422927 0.77 RXRA (0.70) RXRARARBRARGRXRBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000059861-A1 SELECTIVE RETINOIC ACID ANALOGS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-10-12 WO disclosed