SCHEMBL8028109

SCHEMBL8028109

Fc1ccc2c(c1)-n1nnc(-c3ccccc3)c1CNC2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
DHODH Q02127 3/20 0.36
MAP2K4 P45985 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
DCTPP1 Q9H773 1/20 0.34
SIGMAR1 Q99720 4/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP3A4 P08684 1/20 0.33
TP53 P04637 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996189 0.92 CYP1A2 (0.39) NPC1RAB9ADHODHCYP1A2CYP2D6
SCHEMBL14996193 0.90 NPC1 (0.50) NPC1RAB9ADHODHMAP2K4SMN1; SMN2
SCHEMBL8033819 0.86 NPC1 (0.42) NPC1RAB9ADHODHSMN1; SMN2DCTPP1
SCHEMBL8019842 0.85 POLB (0.39) NPC1RAB9ACYP1A2CYP2D6TP53
SCHEMBL14996188 0.85 NPC1 (0.38) NPC1RAB9ADHODHSMN1; SMN2CYP1A2
SCHEMBL8020266 0.84 NPC1 (0.40) NPC1RAB9ADHODHSMN1; SMN2CYP3A4
SCHEMBL8029354 0.84 KCNN4 (0.38) NPC1RAB9ASMN1; SMN2TP53HTR2B
SCHEMBL13002498 0.83 NPC1 (0.39) NPC1RAB9ADHODHDCTPP1CYP1A2
SCHEMBL8028113 0.82 NPC1 (0.40) NPC1RAB9ADHODHCYP1A2CYP2D6
SCHEMBL8033068 0.81 NPC1 (0.37) NPC1RAB9ADHODHCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
WO-2009093269-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LIMITED (IN) 2009-07-30 WO disclosed