SCHEMBL8028113

SCHEMBL8028113

Fc1ccc(-c2nnn3c2CNCc2cc(F)ccc2-3)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
DHODH Q02127 3/20 0.34
ESR1 P03372 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996193 0.92 NPC1 (0.50) NPC1RAB9ADHODH
SCHEMBL8033071 0.90 LMNA (0.39) NPC1RAB9A
SCHEMBL14996189 0.90 CYP1A2 (0.39) NPC1RAB9ACYP1A2CYP2D6DHODH
SCHEMBL8033068 0.88 NPC1 (0.37) NPC1RAB9ACYP1A2CYP2D6DHODH
SCHEMBL14996188 0.87 NPC1 (0.38) NPC1RAB9ACYP1A2CYP2D6DHODH
SCHEMBL8028109 0.82 NPC1 (0.47) NPC1RAB9ACYP1A2CYP2D6DHODH
SCHEMBL8031216 0.81 KCNN4 (0.38) NPC1RAB9A
SCHEMBL13059497 0.81 ADORA2A (0.39) NPC1RAB9ADHODH
SCHEMBL13002540 0.81 NPC1 (0.41) NPC1RAB9ADHODH
SCHEMBL8019842 0.80 POLB (0.39) NPC1RAB9ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
WO-2009093269-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LIMITED (IN) 2009-07-30 WO disclosed