SCHEMBL8028173

SCHEMBL8028173

CCOC(=O)CCCCn1c(Cc2ccc(C#N)cc2)nc2cc(N(C)C(=O)C3CCCCC3)ccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 20/20 0.59
CSNK1D P48730 4/20 0.58
RPS6KA3 P51812 4/20 0.58
DYRK1A Q13627 4/20 0.58
AURKB Q96GD4 4/20 0.58
IRAK4 Q9NWZ3 4/20 0.58
CHEK2 O96017 3/20 0.58
PRKCG P05129 3/20 0.58
MAP4K4 O95819 3/20 0.58
PHKG2 P15735 3/20 0.58
MARK3 P27448 3/20 0.58
CSNK1A1 P48729 3/20 0.58
CLK2 P49760 3/20 0.58
IRAK1 P51617 3/20 0.58
NEK4 P51957 3/20 0.58
CSNK1G2 P78368 3/20 0.58
MAP4K2 Q12851 3/20 0.58
CAMK2G Q13555 3/20 0.58
PKN2 Q16513 3/20 0.58
SRPK1 Q96SB4 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028166 0.98 ITK (0.59) ITKCSNK1DRPS6KA3DYRK1AAURKB
Hydrochloric Acid SCHEMBL8028490 0.87 ITK (0.50) ITKCSNK1DRPS6KA3DYRK1AAURKB
SCHEMBL8028272 0.85 CNR2 (0.60) ITKCSNK1DRPS6KA3DYRK1AAURKB
Hydrochloric Acid SCHEMBL8031513 0.85 ITK (0.51) ITKCSNK1DRPS6KA3DYRK1AAURKB
SCHEMBL8030096 0.85 NPC1 (0.47) ITKCSNK1DRPS6KA3DYRK1AAURKB
SCHEMBL8026960 0.78 CNR2 (0.51) ITK
SCHEMBL8028171 0.77 CNR2 (0.44) ITK
Hydrochloric Acid SCHEMBL8027379 0.77 ITK (0.53) ITKCSNK1DRPS6KA3DYRK1AAURKB
SCHEMBL8026447 0.75 F2 (0.41)
SCHEMBL8016086 0.75 ITK (0.42) ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060166-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS Boehringer Ingelheim Pharma KG (DE) 2000-12-20 EP disclosed
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed
WO-1999040072-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-08-12 WO disclosed