SCHEMBL8028228

SCHEMBL8028228

C[Si](C)(C)CCOCn1cnc2cc(CCO)cnc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
DGAT1 O75907 2/20 0.38
USP2 O75604 1/20 0.34
PNP P00491 1/20 0.34
TSHR P16473 1/20 0.34
EDNRA P25101 1/20 0.34
HTR2A P28223 1/20 0.34
RECQL P46063 1/20 0.34
BLM P54132 1/20 0.34
HBB P68871 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CSF1R P07333 5/20 0.32
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19538828 0.81 BRD4 (0.46) BRD4CREBBPDGAT1CSF1RMEN1
SCHEMBL29868688 0.80 BRD4 (0.46) BRD4CREBBPDGAT1USP2PNP
SCHEMBL189854 0.80 BRD4 (0.46) BRD4CREBBPDGAT1HSD17B10CSF1R
SCHEMBL19531663 0.78 BRD4 (0.44) BRD4CREBBPDGAT1CSF1RNTRK1
SCHEMBL8014137 0.78 BRD4 (0.44) BRD4CREBBPDGAT1
SCHEMBL17457845 0.77 BRD4 (0.44) BRD4CREBBPDGAT1CSF1R
SCHEMBL29600164 0.75 BRD4 (0.43) BRD4CREBBPDGAT1
SCHEMBL15183831 0.75 BRD4 (0.43) BRD4CREBBPDGAT1
SCHEMBL8012052 0.75 BRD4 (0.41) BRD4CREBBPDGAT1CSF1RNTRK1
SCHEMBL8012757 0.75 BRD4 (0.47) BRD4CREBBPCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6110931-A FOR PREGNANCY PROPHYLAXIS AND TREATMENT OF GLANDULAR DISORDERS, HORMONE DEFICIENCY DISORDERS, GASTROINTESTINAL DISORDERS, GROWTH DISORDERS MERCK & CO., INC. (US) 2000-08-29 US disclosed
US-6025366-A Antagonists of gonadotropin releasing hormone MERCK & CO., INC. (US) 2000-02-15 US disclosed