SCHEMBL8028571

SCHEMBL8028571

Cc1coc(C(C)C#Cc2ccccc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
THPO P40225 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRM1 Q13255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11557712 0.71 HDAC1 (0.36) GRM5KDM4EMEN1KMT2AHDAC6
Benzene SCHEMBL7220483 0.69
SCHEMBL30172156 0.68 APP (0.48) GRM5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL8028575 0.68 GRM5 (0.46) GRM5NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL28242920 0.66 APP (0.50) GRM5NPC1RAB9AKDM4EALDH1A1
SCHEMBL3031415 0.65 APP (0.55) GRM5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL20773694 0.65 TAAR1 (0.48) SMN1; SMN2HDAC6HTR2A
SCHEMBL23866038 0.64
SCHEMBL31727818 0.64
SCHEMBL2554839 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037367-A Substituted-pent-4-ynoic acids SMITHKLINE BEECHAM CORPORATION (US) 2000-03-14 US claimed