SCHEMBL8028575

SCHEMBL8028575

Cc1coc(CCC#Cc2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.46
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
THPO P40225 2/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
CYP2D6 P10635 1/20 0.38
PKM P14618 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11557714 0.74 NPC1 (0.45) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL5249356 0.70 FFAR1 (0.66) GRM5FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL4285196 0.70 ATM (0.44) CYP2D6
SCHEMBL7220481 0.69 L3MBTL1 (0.44) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL11453485 0.68 SMN1; SMN2 (0.42) NPC1RAB9ASMN1; SMN2MEN1ALDH1A1
SCHEMBL8028571 0.68 GRM5 (0.39) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL10768214 0.68 CYP1A2 (0.64) GRM5FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL10798421 0.67 FFAR1 (0.61) GRM5FFAR1FFAR4NPC1SMN1; SMN2
SCHEMBL10233436 0.66 CYP1A2 (0.47) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL21894058 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037367-A Substituted-pent-4-ynoic acids SMITHKLINE BEECHAM CORPORATION (US) 2000-03-14 US claimed