SCHEMBL8028803

SCHEMBL8028803

Fc1ccc2c(c1)-n1c(nnc1-c1ccccc1)CNC2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
TSHR P16473 1/20 0.38
P2RX7 Q99572 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
AVPR1A P37288 2/20 0.35
HPGD P15428 1/20 0.35
AKT1 P31749 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13002472 0.84 TSHR (0.52) CYP17A1CYP3A4CYP19A1CYP11B1CYP11B2
SCHEMBL13002467 0.81 CYP11B2 (0.41) CYP11B1CYP11B2CYP1A2CYP2D6AVPR1A
SCHEMBL14996186 0.75 CYP11B2 (0.42) CYP11B2CYP1A2CYP2D6AVPR1A
SCHEMBL3760445 0.72 AVPR1A (0.32) AVPR1A
SCHEMBL14996183 0.69 CYP11B2 (0.38) CYP11B1CYP11B2CYP1A2CYP2D6AVPR1A
SCHEMBL13002490 0.68 S1PR1 (0.35) CYP3A4CYP1A2CYP2D6HPGDNPC1
SCHEMBL8028802 0.66 BRD4 (0.50) CYP11B1CYP11B2TSHRAVPR1AHPGD
SCHEMBL12841365 0.66 TSHR (0.62) CYP17A1CYP3A4CYP19A1CYP11B1CYP11B2
SCHEMBL12841355 0.66 TSHR (0.50) CYP17A1CYP3A4CYP19A1CYP11B1CYP11B2
Trifluoroacetic Acid SCHEMBL3760442 0.66 CYP11B1 (0.34) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC PHARMA LIMITED (IN) 2010-12-09 US disclosed
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC PHARMA LIMITED (IN) 2010-12-09 US disclosed
WO-2009093269-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LIMITED (IN) 2009-07-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS DPP4, DPP3, DPP8 CYP17A1 1100/4885CYP3A4 8/4885CYP19A1 1064/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.