SCHEMBL8030637

SCHEMBL8030637

COc1cccc(P(c2ccccc2)c2cccc(OC)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA4 P22748 1/20 0.52
CYP3A4 P08684 3/20 0.50
TDP1 Q9NUW8 1/20 0.50
ACHE P22303 1/20 0.48
MAOB P27338 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LTA4H P09960 1/20 0.45
CYP1A2 P05177 2/20 0.43
CYP2A6 P11509 1/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ENPP2 Q13822 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
LMNA P02545 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676480 1.00 CA4 (0.52) CA4CYP3A4TDP1ACHEMAOB
SCHEMBL29635198 0.94 ACHE (0.54) CA4CYP3A4ACHECA1CA2
SCHEMBL197286 0.94 ACHE (0.54) CA4CYP3A4ACHECA1CA2
1,3-Dimethoxybenzene SCHEMBL28127772 0.92 CA4 (0.52) CA4CYP3A4TDP1ACHEMAOB
SCHEMBL5713343 0.91 ACHE (0.52) CA4CYP3A4ACHECA1CA2
Phosphine SCHEMBL6466867 0.91 ACHE (0.52) CA4CYP3A4ACHECA1CA2
Hydrochloric Acid SCHEMBL5427158 0.91 ACHE (0.52) CA4CYP3A4ACHECA1CA2
1,3-Dimethoxybenzene SCHEMBL28127423 0.90 MAOB (0.50) CA4CYP3A4TDP1ACHEMAOB
SCHEMBL16487759 0.86 ACHE (0.69) CA4CYP3A4ACHEMAOBCA1
SCHEMBL20873235 0.86 ACHE (0.47) CA4CYP3A4ACHEMAOBCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984909-A1 USE OF A RHODIUM CATALYST FOR HYDROAMINATION AND/OR OXIDATIVE AMINATION OF ARYL-SUBSTITUTED OLEFINS AND METHOD FOR PRODUCING A 2-ARYL VINYL AMINE Aventis Research & Technologies GmbH & Co KG (DE) 2000-03-15 EP claimed
WO-1998054115-A1 USE OF A RHODIUM CATALYST FOR HYDROAMINATION AND/OR OXIDATIVE AMINATION OF ARYL-SUBSTITUTED OLEFINS AND METHOD FOR PRODUCING A 2-ARYL VINYL AMINE AVENTIS RESEARCH & TECHNOLOGIES GMBH & (DE) 1998-12-03 WO claimed
EP-0984909-A1 USE OF A RHODIUM CATALYST FOR HYDROAMINATION AND/OR OXIDATIVE AMINATION OF ARYL-SUBSTITUTED OLEFINS AND METHOD FOR PRODUCING A 2-ARYL VINYL AMINE Aventis Research & Technologies GmbH & Co KG (DE) 2000-03-15 EP disclosed
WO-1998054115-A1 USE OF A RHODIUM CATALYST FOR HYDROAMINATION AND/OR OXIDATIVE AMINATION OF ARYL-SUBSTITUTED OLEFINS AND METHOD FOR PRODUCING A 2-ARYL VINYL AMINE AVENTIS RESEARCH & TECHNOLOGIES GMBH & (DE) 1998-12-03 WO disclosed
EP-0271145-B1 PROCESS FOR THE CARBONYLATION OF CONJUGATED DIENES SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-08-21 EP disclosed
US-4824817-A Catalyst for the carbonylation of conjugated dienes SHELL OIL COMPANY (US) 1989-04-25 US disclosed
EP-0271145-A2 Process for the carbonylation of conjugated dienes SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1988-06-15 EP disclosed