SCHEMBL8031472

SCHEMBL8031472

C=C(N)c1ccc(SCC(NC(=O)CCC(N)C(=O)O)C(=O)O)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL858566 0.92 ALDH1A1 (0.51) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL13868150 0.90 PTGS1 (0.47) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL13868159 0.85 APEX1 (0.48) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL13295134 0.84 ALDH1A1 (0.45) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20856994 0.83 PTGS1 (0.48) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL858563 0.83 PTGS1 (0.48) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL859188 0.81 SMN1; SMN2 (0.44) APEX1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1524585 0.77 PTGS1 (0.50) ALDH1A1MAPT
SCHEMBL13157335 0.77 PTGS1 (0.50) ALDH1A1MAPT
SCHEMBL1524589 0.77 PTGS1 (0.50) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012454-A1 METHODS OF TREATING METASTATIC BREAST CANCER WITH 4-IODO-3-NITROBENZAMIDE AND IRINOTECAN BIPAR SCIENCES, INC. (US) 2012-01-26 WO disclosed
WO-2009073869-A1 TREATMENT OF CANCER WITH COMBINATIONS OF TOPOISOMERASE INHIBITORS AND PARP INHIBITORS BIPAR SCIENCES, INC. (US) 2009-06-11 WO disclosed