Pyrimidine

Pyrimidine

SCHEMBL8031985

CCCNC1CCNCC1.c1cncnc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNAI3 P08754 3/20 0.51
GNAO1 P09471 3/20 0.51
GNAI1 P63096 3/20 0.51
SOS1 Q07889 1/20 0.43
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
KCNH2 Q12809 1/20 0.38
KDM1A O60341 1/20 0.35
CYP1A2 P05177 2/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
EPHX1 P07099 1/20 0.35
PIM1 P11309 1/20 0.34
DRD3 P35462 6/20 0.33
DRD2 P14416 5/20 0.33
AXL P30530 1/20 0.33
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrimidine SCHEMBL7658961 0.86 KCNH2 (0.53) GNAI3GNAO1GNAI1SOS1ROCK2
SCHEMBL1197783 0.84 GNAI3 (0.68) GNAI3GNAO1GNAI1SOS1KCNH2
Pyrimidine SCHEMBL8028462 0.77 KDM1A (0.40) SOS1ROCK2ROCK1KCNH2KDM1A
SCHEMBL4979028 0.72
SCHEMBL1070277 0.72 GNAI3 (0.81) GNAI3GNAO1GNAI1SOS1KCNH2
SCHEMBL5761715 0.72
SCHEMBL18711243 0.72
SCHEMBL3265058 0.71 GNAI3 (0.92) GNAI3GNAO1GNAI1SOS1KCNH2
SCHEMBL19604164 0.69 GNAI3 (0.96) GNAI3GNAO1GNAI1KCNH2EPHX1
SCHEMBL7319928 0.69 GNAI3 (0.96) GNAI3GNAO1GNAI1KCNH2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000059498-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed