SCHEMBL8034148

SCHEMBL8034148

COc1ccc2nc(C=Cc3nc4ccccc4s3)sc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.60
MEN1 O00255 7/20 0.60
KMT2A Q03164 7/20 0.60
MAPT P10636 6/20 0.60
KDM4E B2RXH2 4/20 0.60
ALDH1A1 P00352 3/20 0.60
POLB P06746 2/20 0.60
GAA P10253 1/20 0.60
HTT P42858 1/20 0.60
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C19 P33261 1/20 0.55
ATP4A P20648 5/20 0.54
ATP4B P51164 5/20 0.54
PDK1 Q15118 1/20 0.54
TDP1 Q9NUW8 3/20 0.54
SMN1; SMN2 Q16637 7/20 0.53
NPC1 O15118 4/20 0.53
NFKB1 P19838 3/20 0.53
NFKB2 Q00653 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24157673 0.87 CYP1A2 (0.56) RAB9AMEN1KMT2AMAPTHTT
SCHEMBL825345 0.85 MEN1 (0.66) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL825346 0.85 MEN1 (0.66) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL13936229 0.85 ATP4A (0.66) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL6493241 0.84 MEN1 (0.70) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL6493243 0.84 MEN1 (0.70) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL8031699 0.83 MAPT (0.49) RAB9AMEN1KMT2AMAPTKDM4E
SCHEMBL6115945 0.82 ATP4A (0.49) RAB9AMEN1KMT2AMAPTALDH1A1
SCHEMBL6115942 0.82 ATP4A (0.49) RAB9AMEN1KMT2AMAPTALDH1A1
SCHEMBL12545463 0.80 CYP1A2 (0.59) RAB9AMEN1KMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6140051-A USE IN THE FIELD OF BIOLOGICAL ASSAYS PROMEGA BIOSCIENCES, INC. (US) 2000-10-31 US disclosed
EP-1000042-A1 FLUORESCENT DIBENZAZOLE DERIVATIVES AND METHODS RELATED THERETO Promega Biosciences, Inc. (US) 2000-05-17 EP disclosed
WO-2000004007-A1 FLUORESCENT DIBENZAZOLE DERIVATIVES AND METHODS RELATED THERETO PROMEGA BIOSCIENCES, INC. (US) 2000-01-27 WO disclosed
WO-1999003849-A1 FLUORESCENT DIBENZAZOLE DERIVATIVES AND METHODS RELATED THERETO PROMEGA BIOSCIENCES, INC. (US) 1999-01-28 WO disclosed