SCHEMBL8034393

SCHEMBL8034393

Brc1nc(Sc2nnc(-c3ccccc3)s2)sc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.48
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.38
PKM P14618 2/20 0.37
ATM Q13315 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA5A P35218 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GSK3B P49841 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TERT O14746 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TNF P01375 1/20 0.32
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042113 0.82 HDAC6 (0.43) HDAC6ALDH1A1POLBPKMATM
SCHEMBL8050088 0.78 KDM4E (0.45) ALDH1A1PKMMEN1KMT2ANPC1
SCHEMBL8042376 0.78 ALDH1A1 (0.45) HDAC6ALDH1A1POLBMEN1KMT2A
SCHEMBL8042760 0.77 ATM (0.47) ALDH1A1POLBATMMEN1KMT2A
SCHEMBL8048725 0.76 ALDH1A1 (0.53) HDAC6ALDH1A1POLBATMKMT2A
SCHEMBL28353372 0.75 HDAC6 (0.64) HDAC6ALDH1A1POLBPKMATM
SCHEMBL8050637 0.74 HDAC6 (0.49) HDAC6ALDH1A1POLBPKMMEN1
SCHEMBL8034279 0.73 HDAC6 (0.45) HDAC6ALDH1A1POLBPKMATM
SCHEMBL14832839 0.73 ALDH1A1 (0.43) ALDH1A1POLBPKMMEN1KMT2A
SCHEMBL8045096 0.71 PDPK1 (0.51) HDAC6ALDH1A1POLBPKMATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed