SCHEMBL8034773

SCHEMBL8034773

C/C=C/[C@H]1CC[C@H](C2CCC(c3cnc(-c4ccc(F)c(F)c4)nc3)CC2)CC1

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
HDAC4 P56524 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP11B2 P19099 1/20 0.31
OPRL1 P41146 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
DHODH Q02127 1/20 0.30
RXRA P19793 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378335 0.96 PDGFRB (0.33) ACACBPDGFRBPDGFRAHDAC4CYP17A1
SCHEMBL9312598 0.96 PDGFRB (0.33) ACACBPDGFRBPDGFRAHDAC4CYP17A1
SCHEMBL8378334 0.96 PDGFRB (0.33) ACACBPDGFRBPDGFRAHDAC4CYP17A1
SCHEMBL8382748 0.85 CYP11B1 (0.34) ACACBHDAC4CYP11B2DHODHRXRA
SCHEMBL8383601 0.85 S1PR1 (0.36) CYP11B2DHODH
SCHEMBL8383609 0.85 S1PR1 (0.36) CYP11B2DHODH
SCHEMBL9313247 0.85 CYP11B1 (0.34) ACACBHDAC4CYP11B2DHODHRXRA
SCHEMBL9312273 0.85 S1PR1 (0.36) CYP11B2DHODH
SCHEMBL8382750 0.85 CYP11B1 (0.34) ACACBHDAC4CYP11B2DHODHRXRA
SCHEMBL8024912 0.85 CYP17A1 (0.33) CYP17A1CYP3A4CYP11B2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497176-B1 Four rings compounds and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 2000-04-05 EP disclosed
EP-0497176-A2 Four rings compounds and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1992-08-05 EP disclosed