Lysine

Lysine

SCHEMBL8039281

NCCCC[C@H](N)C(=O)O.O=Cc1ccccc1O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.56
TRIM24 O15164 1/20 0.50
TRIM33 Q9UPN9 1/20 0.50
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
DPP8 Q6V1X1 1/20 0.44
DPP9 Q86TI2 1/20 0.44
DPP7 Q9UHL4 1/20 0.44
MMP2 P08253 1/20 0.43
ARG2 P78540 4/20 0.41
ARG1 P05089 3/20 0.41
KIF11 P52732 4/20 0.40
LTA4H P09960 1/20 0.39
NOS1 P29475 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL8039288 1.00 GSR (0.56) GSRTRIM24TRIM33POLBKMT2A
Lysine SCHEMBL28249818 0.87 GSR (0.69) GSRPOLBKMT2ATDP1DPP8
Lysine SCHEMBL28249816 0.87 GSR (0.69) GSRPOLBKMT2ATDP1DPP8
Salicyladehyde SCHEMBL8035802 0.84 TRIM24 (0.58) TRIM24TRIM33KMT2ATDP1KIF11
Salicyladehyde SCHEMBL8035808 0.84 TRIM24 (0.58) TRIM24TRIM33KMT2ATDP1KIF11
2-Methoxybenzaldehyde SCHEMBL8039080 0.82 GRIK1 (0.51) GSRPOLBKMT2ATDP1DPP8
2-Methoxybenzaldehyde SCHEMBL8039077 0.82 GRIK1 (0.51) GSRPOLBKMT2ATDP1DPP8
Lysine SCHEMBL9643349 0.81 GSR (0.61) GSRPOLBKMT2ATDP1DPP8
Lysine SCHEMBL1649467 0.80 GSR (0.59) GSRPOLBKMT2ATDP1DPP8
Lysine SCHEMBL1650193 0.80 GSR (0.59) GSRPOLBKMT2ATDP1DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
US-3957760-A AMINO ACID DERIVATIVES E. R. SQUIBB & SONS, INC. (US) 1976-05-18 US disclosed