Lysine

Lysine

SCHEMBL1649467

NCCCC[C@H](N)C(=O)O.O=C(O)c1ccccc1O

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.59
KDM4E B2RXH2 2/20 0.53
CA12 O43570 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
HMGB1 P09429 1/20 0.53
HPGD P15428 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA7 P43166 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CA9 Q16790 1/20 0.53
NAPRT Q6XQN6 1/20 0.53
CA14 Q9ULX7 1/20 0.53
TDP1 Q9NUW8 2/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.47
DPP8 Q6V1X1 1/20 0.46
DPP9 Q86TI2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL1650193 1.00 GSR (0.59) GSRKDM4ECA12ALDH1A1CA1
Lysine SCHEMBL17965939 0.99 GSR (0.57) GSRKDM4ECA12ALDH1A1CA1
Lysine SCHEMBL17965940 0.99 GSR (0.57) GSRKDM4ECA12ALDH1A1CA1
Phthalic Acid SCHEMBL19210211 0.91 GSR (0.67) GSRALDH1A1TDP1POLBKMT2A
Phthalic Acid SCHEMBL19210210 0.91 GSR (0.67) GSRALDH1A1TDP1POLBKMT2A
Lysine SCHEMBL28249816 0.89 GSR (0.69) GSRTDP1POLBKMT2ADPP8
Lysine SCHEMBL28249818 0.89 GSR (0.69) GSRTDP1POLBKMT2ADPP8
Aspirin SCHEMBL4094492 0.87 KDM4E (0.53) GSRKDM4ECA12ALDH1A1CA1
Lysine SCHEMBL28275800 0.85 GSR (0.59) GSRTDP1POLBKMT2ADPP8
Salicylic Acid SCHEMBL28307845 0.85 ALDH1A1 (0.50) KDM4ECA12ALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115607556-A Medicine for preventing and treating asthma, chronic obstructive pulmonary disease, allergic diseases, etc 刘力 2023-01-17 CN claimed
WO-2013020527-A1 UTILIZATION OF ALAPTIDE AS TRANSDERMAL PENETRATION MODIFIER IN PHARMACEUTICAL COMPOSITIONS FOR HUMAN AND VETERINARY APPLICATIONS CONTAINING ANTI-INFLAMMATORY DRUGS AND/OR ANTIMICROBIAL CHEMOTHERAPEUTICS UNIVERSITY OF VETERINARY AND PHARMACEUTICAL SCIENCES BRNO FACULTY OF PHARMACY (CZ) 2013-02-14 WO claimed
US-4988683-A Administering lysine acetylsalicylate by mouth for pain and hypothermia CORBIERE JEROME (FR) 1991-01-29 US claimed
US-20250049674-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST A MEROCYANINE AND A HYDROTROPE L'OREAL (FR) 2025-02-13 US disclosed
US-20250025393-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING A MEROCYANINE AND DIPROPYLENE GLYCOL L'OREAL (FR) 2025-01-23 US disclosed
US-20250009625-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING A MEROCYANINE AND AT LEAST ONE DIOL COMPRISING FROM 4 TO 7 CARBON ATOMS L'OREAL (FR) 2025-01-09 US disclosed
US-20240423888-A1 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST ONE MEROCYANINE AND AT LEAST ASCORBIC ACID AND/OR A DERIVATIVE THEREOF L'OREAL (FR) 2024-12-26 US disclosed
CN-118871078-A Cosmetic or dermatological composition comprising at least a merocyanine and a hydrotrope 欧莱雅 2024-10-29 CN disclosed
EP-4447895-A1 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST ONE MEROCYANINE AND AT LEAST ASCORBIC ACID AND/OR A DERIVATIVE THEREOF L'OREAL (FR) 2024-10-23 EP disclosed
CN-118804735-A Cosmetic and/or dermatological composition comprising at least one merocyanine and at least ascorbic acid and/or derivatives thereof 莱雅公司 2024-10-18 CN disclosed
CN-118678942-A Cosmetic or dermatological composition comprising a merocyanine and at least one glycol comprising 4 to 7 carbon atoms 莱雅公司 2024-09-20 CN disclosed
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed
CN-1468104-A Use of a combination of purine activity and AINS activity for the preparation of an antithrombotic or antiinflammatory agent ����ŵ÷�¹�˾ 2004-01-14 CN disclosed
EP-0936899-A4 COSMETIC COMPOSITIONS PROCTER & GAMBLE (US) 2002-01-02 EP disclosed
US-6267978-B1 COSMETIC FOR REGULATION OF THE OILY AND/OR SHINY APPEARANCE OF SKIN THE PROCTER & GAMBLE COMPANY 2001-07-31 US disclosed
US-6143310-A WATER IN OIL EMULSION CONTAINING AMINO ACID SALT OF SALICYLIC ACID THE PROCTER & GAMBLE COMPANY (US) 2000-11-07 US disclosed
EP-0936899-A1 COSMETIC COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1999-08-25 EP disclosed
WO-1998010741-A1 COSMETIC COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1998-03-19 WO disclosed
WO-1996024331-A1 NEW MEDICAL FORMS WITH PROLONGED EFFECT APPLIED IN EYE MEDICINE AND THE METHOD FOR PREPARATION THEREOF ÚSTAV MAKROMOLEKULÁRNÍ CHEMIE AKADEMIE VE^¿D C^¿ESKÉ REPUBLIKY (CZ) 1996-08-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250009625-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING A MEROCYANINE AND AT LEAST ONE DIOL COMPRISING FROM 4 TO 7 CARBON ATOMS KRT18, DSC1, ECH1 GSR 3097/4885KDM4E 2121/4885CA12 141/4885
US-20240423888-A1 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST ONE MEROCYANINE AND AT LEAST ASCORBIC ACID AND/OR A DERIVATIVE THEREOF KRT18, PROC, DSC1 GSR 1290/4885KDM4E 1082/4885CA12 547/4885
US-20250049674-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST A MEROCYANINE AND A HYDROTROPE NAPRT, NAMPT, NNMT GSR 2121/4885KDM4E 2686/4885CA12 961/4885
US-20250025393-A1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING A MEROCYANINE AND DIPROPYLENE GLYCOL KRT18, DSC1, DSG1 GSR 3344/4885KDM4E 1786/4885CA12 50/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.