SCHEMBL8039359

SCHEMBL8039359

[c]1n[nH]cc1N1CCCc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.42
JAK2 O60674 2/20 0.41
JAK3 P52333 1/20 0.41
PTK2 Q05397 1/20 0.41
NUDT1 P36639 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 5/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 2/20 0.38
TSHR P16473 2/20 0.38
STAT3 P40763 1/20 0.38
NOTUM Q6P988 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3422889 0.75 ROCK1 (0.49) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL3145069 0.72 ROCK1 (0.46) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL11199183 0.70 ROCK1 (0.43) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL4431357 0.69 ROCK1 (0.56) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL29478502 0.69 ROCK1 (0.51) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL693233 0.69 ROCK1 (0.51) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL5245431 0.68 ROCK1 (0.63) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL17486069 0.68 JAK2 (0.53) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL11880068 0.67 ROCK1 (0.50) ROCK1L3MBTL1JAK2JAK3PTK2
SCHEMBL10621398 0.67 ROCK1 (0.54) ROCK1L3MBTL1JAK2JAK3PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000066562-A1 PYRAZOLES HAVING ANTIINFLAMMATORY ACTIVITY DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-11-09 WO claimed
WO-2000066562-A1 PYRAZOLES HAVING ANTIINFLAMMATORY ACTIVITY DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-11-09 WO disclosed