SCHEMBL8039486

SCHEMBL8039486

N[C@H](Cc1ccc(-c2ccccc2O)nc1)NC(=O)[C@@H]1CCCCN1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSC P53634 7/20 0.46
CTSK P43235 3/20 0.41
KCNH2 Q12809 2/20 0.41
CCNT1 O60563 1/20 0.38
CDK1 P06493 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38
MNAT1 P51948 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
GHSR Q92847 6/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1499022 0.86 CTSC (0.65) CTSCCTSKKCNH2
SCHEMBL1499017 0.86 CTSC (0.65) CTSCCTSKKCNH2
SCHEMBL8037816 0.83 CTSC (0.47) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8038040 0.82 CTSC (0.46) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8031912 0.77 CTSC (0.56) CTSCCTSKKCNH2CYP3A4CYP2D6
SCHEMBL8039150 0.75 CTSC (0.59) CTSCCTSKKCNH2CYP3A4CYP2D6
SCHEMBL8031916 0.75 CTSC (0.54) CTSCCTSKKCNH2CYP3A4CYP2D6
SCHEMBL8040349 0.74 CTSC (0.66) CTSCCTSKKCNH2CYP3A4CYP2D6
SCHEMBL8041660 0.73 CTSC (0.48) CTSCCTSKKCNH2CYP3A4CYP2D6
SCHEMBL3658702 0.73 CTSC (0.44) CTSCCTSKKCNH2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed