SCHEMBL8037816

SCHEMBL8037816

Nc1ccc(-c2ccc(C[C@@H](N)NC(=O)[C@@H]3CCCCN3)cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSC P53634 8/20 0.47
CTSK P43235 3/20 0.47
KCNH2 Q12809 2/20 0.47
SCN3A Q9NY46 2/20 0.40
SCN9A Q15858 1/20 0.40
ATR Q13535 1/20 0.38
TPH1 P17752 1/20 0.38
HTR2C P28335 2/20 0.37
HTR2B P41595 1/20 0.37
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
ULK1 O75385 1/20 0.36
BRAF P15056 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8038040 0.91 CTSC (0.46) CTSCCTSKKCNH2SCN3ASCN9A
SCHEMBL8039486 0.83 CTSC (0.46) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8039150 0.79 CTSC (0.59) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL12422470 0.78 CTSC (0.79) CTSCCTSKKCNH2
SCHEMBL8039004 0.78 CTSC (0.58) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8039503 0.78 CTSC (0.51) CTSCCTSKKCNH2SCN3ASCN9A
SCHEMBL8023034 0.77 CTSC (0.52) CTSCCTSKKCNH2SCN3ASCN9A
SCHEMBL8036103 0.77 CTSC (0.60) CTSCCTSKKCNH2
SCHEMBL8040349 0.76 CTSC (0.66) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8036119 0.76 CTSC (0.55) CTSCCTSKKCNH2HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed