SCHEMBL8041279

SCHEMBL8041279

Cc1ccc2c(c1)c1c(n2CC(O)c2ccccc2)CCNC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.51
GRIN2D O15399 2/20 0.49
GRIN3B O60391 2/20 0.49
GRIN1 Q05586 2/20 0.49
GRIN2A Q12879 2/20 0.49
GRIN2B Q13224 2/20 0.49
GRIN2C Q14957 2/20 0.49
GRIN3A Q8TCU5 2/20 0.49
SIRT1 Q96EB6 1/20 0.49
LMNA P02545 2/20 0.47
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
BCHE P06276 2/20 0.46
KDM4E B2RXH2 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
ADRA2A P08913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12480649 0.89 SIRT2 (0.47) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12480358 0.88 SIRT2 (0.46) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL15132910 0.87 SIRT2 (0.46) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL16709561 0.83 KMT2A (0.51) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3229857 0.81 GRIN2D (0.64) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL16900206 0.81 KMT2A (0.45) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3032023 0.80 GRIN1 (0.75) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3722443 0.80 HRH1 (0.67) SIRT2GRIN1GRIN2AGRIN2BSIRT1
SCHEMBL16140204 0.80 SIRT2 (0.60) SIRT2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL16140207 0.79 SIRT2 (0.59) SIRT2GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009082268-A2 LIGANDS OF α-ADRENOCEPTORS AND OF DOPAMINE, HISTAMINE, IMIDAZOLINE AND SEROTONIN RECEPTORS AND THE USE THEREOF ALLA CHEM, LLC (US) 2009-07-02 WO disclosed