SCHEMBL8041370

SCHEMBL8041370

CC(C)(C1CCN(C(=O)c2ccccc2CC(F)(F)F)CC1)S(=O)(=O)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 12/20 0.55
CYP3A4 P08684 2/20 0.55
NR1I2 O75469 2/20 0.49
AKR1C3 P42330 1/20 0.41
HSD11B1 P28845 1/20 0.41
MGLL Q99685 1/20 0.40
PKLR P30613 1/20 0.40
SCN9A Q15858 1/20 0.40
RORC P51449 1/20 0.40
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
CFD P00746 1/20 0.38
KLK7 P49862 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044492 0.90 CACNA1B (0.54) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3025486 0.87 CACNA1B (0.65) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3038986 0.84 CACNA1B (0.56) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3032278 0.84 CACNA1B (0.59) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3031674 0.80 CACNA1B (0.76) CACNA1BCYP3A4NR1I2HSD11B1SCN9A
SCHEMBL3035644 0.80 CACNA1B (0.82) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3035386 0.80 HSD11B1 (0.57) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3032252 0.80 CACNA1B (0.54) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3038099 0.80 CACNA1B (0.61) CACNA1BCYP3A4NR1I2AKR1C3HSD11B1
SCHEMBL3025452 0.80 CACNA1B (0.70) CACNA1BCYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO disclosed