SCHEMBL8042853

SCHEMBL8042853

CC(C)(C1CCN(C(=O)c2ccc(CC(F)F)cc2S(C)(=O)=O)CC1)S(=O)(=O)c1cncc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 19/20 0.54
NR1I2 O75469 10/20 0.54
CYP3A4 P08684 3/20 0.54
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3037966 0.87 CACNA1B (0.54) CACNA1BNR1I2CYP3A4
SCHEMBL3038145 0.84 CACNA1B (0.60) CACNA1BNR1I2CYP3A4
SCHEMBL8044016 0.84 CACNA1B (0.50) CACNA1BNR1I2CYP3A4
SCHEMBL3034886 0.84 CACNA1B (0.54) CACNA1BNR1I2CYP3A4
SCHEMBL14688807 0.79 CACNA1B (0.55) CACNA1BNR1I2CYP3A4
SCHEMBL3038537 0.78 CACNA1B (0.51) CACNA1BNR1I2CYP3A4
SCHEMBL3035462 0.78 CACNA1B (0.78) CACNA1BNR1I2CYP3A4
SCHEMBL3030681 0.76 CACNA1B (0.64) CACNA1BNR1I2CYP3A4
SCHEMBL3035595 0.76 CACNA1B (0.66) CACNA1BNR1I2CYP3A4
SCHEMBL3042236 0.76 CACNA1B (0.68) CACNA1BNR1I2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO disclosed