SCHEMBL8044016

SCHEMBL8044016

CC(C)(C1CCN(C(=O)c2ccc(CC(F)F)cc2S(C)(=O)=O)CC1)S(=O)(=O)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 17/20 0.50
NR1I2 O75469 9/20 0.50
CYP3A4 P08684 3/20 0.50
SLC9A1 P19634 1/20 0.37
MGLL Q99685 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3042977 0.87 CACNA1B (0.50) CACNA1BNR1I2CYP3A4
SCHEMBL3035240 0.84 CACNA1B (0.56) CACNA1BNR1I2CYP3A4
SCHEMBL3035948 0.84 CACNA1B (0.50) CACNA1BNR1I2CYP3A4
SCHEMBL8042853 0.84 CACNA1B (0.54) CACNA1BNR1I2CYP3A4
SCHEMBL3035462 0.74 CACNA1B (0.78) CACNA1BNR1I2CYP3A4
SCHEMBL3123172 0.73 CACNA1B (0.43) CACNA1BNR1I2CYP3A4MGLL
SCHEMBL3042236 0.72 CACNA1B (0.68) CACNA1BNR1I2CYP3A4
SCHEMBL3036257 0.72 CACNA1B (0.74) CACNA1BNR1I2CYP3A4
SCHEMBL3025559 0.72 CACNA1B (0.86) CACNA1BNR1I2CYP3A4
SCHEMBL3039575 0.72 CACNA1B (0.74) CACNA1BNR1I2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO disclosed