SCHEMBL8043003

SCHEMBL8043003

Cc1cc(Nc2ccnc3c2CC[C@@H]3C)ccc1NCCc1c[nH]c2c(C)cccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
PTGS2 P35354 3/20 0.33
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
GLA P06280 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19114338 0.93 PTGS2 (0.31) PTGS2CDK2
SCHEMBL8075495 0.91 HTR2A (0.36) HTR2AMAPTSMN1; SMN2NPSR1HTR1A
SCHEMBL13130737 0.91 HTR2A (0.36) HTR2AMAPTSMN1; SMN2NPSR1HTR1A
SCHEMBL19114334 0.90 PTGS2 (0.30) PTGS2
SCHEMBL15267542 0.83 EGFR (0.33) PTGS2
SCHEMBL19114668 0.83 PTGS2 (0.30) PTGS2
SCHEMBL19114465 0.83 CDK2 (0.33) PTGS2MEN1USP2ALDH1A1CYP1A2
SCHEMBL13258483 0.82 PTGS2 (0.30) PTGS2
SCHEMBL13258435 0.82 PTGS2 (0.36) SMN1; SMN2PTGS2CDK2PTGS1
SCHEMBL15267231 0.82 PTGS2 (0.30) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037308-A1 INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53 JANSSEN PHARMACEUTICA NV (BE) 2009-03-26 WO disclosed