SCHEMBL8043678

SCHEMBL8043678

CCOCc1ccc(NC(=O)c2c[nH]c3c2C(=O)C(C)(C)CC3)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.57
ROCK1 Q13464 1/20 0.57
CFTR P13569 1/20 0.39
CYP26A1 O43174 2/20 0.36
CYP26B1 Q9NR63 2/20 0.36
TP53 P04637 2/20 0.35
NHERF1 O14745 1/20 0.34
KLKB1 P03952 1/20 0.34
RET P07949 5/20 0.34
TRPV1 Q8NER1 1/20 0.34
NAMPT P43490 1/20 0.34
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ABCG2 Q9UNQ0 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
THRB P10828 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5737070 0.90 ROCK2 (0.58) ROCK2ROCK1CFTRCYP26A1CYP26B1
SCHEMBL7396411 0.86 ROCK2 (0.58) ROCK2ROCK1TP53NPC1MAPT
SCHEMBL7398675 0.85 ROCK2 (0.64) ROCK2ROCK1CFTRTP53NPC1
SCHEMBL7395940 0.82 ROCK2 (0.61) ROCK2ROCK1TP53NPC1MAPT
SCHEMBL7369380 0.82 ROCK2 (0.63) ROCK2ROCK1TP53NPC1MAPT
SCHEMBL7397319 0.82 ROCK2 (0.68) ROCK2ROCK1CFTRTP53NPC1
SCHEMBL7392079 0.80 ROCK2 (0.63) ROCK2ROCK1SMN1; SMN2ALDH1A1HTT
SCHEMBL7384260 0.77 ROCK2 (0.57) ROCK2ROCK1CFTRTP53NAMPT
SCHEMBL7399573 0.75 ROCK2 (0.58) ROCK2ROCK1NPC1MAPTRAB9A
SCHEMBL7398250 0.75 ROCK2 (0.55) ROCK2ROCK1TP53NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080873-A Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands NEUROGEN CORPORATION (US) 2000-06-27 US disclosed